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Oral · GLP-1 agonist

Lotiglipron

11 trials in this molecule. Source: ClinicalTrials.gov, as of July 1, 2026.

Trials

11

Active

0

Recruiting

0

Completed

7

Sites

91

Countries

10

Endpoints

392

Composite endpoints

18

Distinct sites and countries across this molecule's trials. A site running several of its trials counts once, matching the map.

Development

Where the program stands

Trials by phase

Phase 1
10
Phase 2
1

Trials by status

Completed
7
Terminated
4

Evidence coverage

What this asset has been measured on

Endpoints grouped into outcome categories, ranked by how often they are measured across this asset's trials.

Safety / tolerability / PK
331
Weight & body composition
26
Glycemic / diabetes
22
Patient-reported / QoL
8
Renal / kidney
5

Most-measured metrics

Top 20 metrics across this asset's endpoints

AUC₀–∞Safety/PK

35

CmaxSafety/PK

28

TmaxSafety/PK

21

Treatment-emergent AEs (any)Safety/PK

18

Half-lifeSafety/PK

18

Body weight, % changeWeight

13

HOMA-IR (insulin sensitivity)Glycemic

8

Waist circumference, changeWeight

4

HbA1c, % changeGlycemic

4

Fasting glucose, changeGlycemic

4

HbA1c, changeGlycemic

4

Serious AEs (any)Safety/PK

4

Discontinuation due to AESafety/PK

4

Documented hypoglycemiaSafety/PK

4

HbA1c <7.0% achievementGlycemic

2

Body weight, absolute change (kg)Weight

1

≥15% weight-loss respondersWeight

1

Trials

Programs for this asset

Every trial for this molecule, with the same search, filters, and sort as the Trials tab.

11 of 11

Asset / PopulationKey I/E criterionEvidence
NCT05579977Trial to Learn About the Study Medicine (PF-07081532) and Rybelsus in People With Type 2 Diabetes and Separately PF-07081532 in People With Obesity

GLP-1 / incretin class catch-all, Lotiglipron, Semaglutide

Obesity / overweight, Type 2 diabetes

BMI ≥23Ph 2Terminated90Jul 20232results
NCT04305587Multiple Escalating Oral Doses Study of PF-07081532 in Adult Participants With Type 2 Diabetes Mellitus

Lotiglipron

Obesity / overweight, Type 2 diabetes

HbA1c 7-10.5%Ph 1Completed2Jul 20211results
NCT05478603A Study to Understand How the Study Medicine (PF-07081532) is Processed in People With Liver Dysfunction

Lotiglipron

Healthy volunteers, Hepatic impairment

BMI 17.5-38Ph 1Completed2Apr 2023results
NCT05510245A Clinical Trial of the Study Medicine (PF-07081532) in People With Diabetes and Kidney Dysfunction

Lotiglipron

Renal impairment, Type 2 diabetes

BMI 17.5-45.4Ph 1Terminated2Jul 2023results
NCT05671653A Study to Evaluate the Effect of the Experimental GLP-1 Drug PF-07081532 on Blood Levels of Common Birth Control Pills, and Drugs Omeprazole and Midazolam, and Effect of GLP-1 Drug Semaglutide on Midazolam Blood Levels in Healthy Adults With Weight in the Obesity Range

Lotiglipron, Semaglutide

Healthy volunteers, Obesity / overweight

BMI 30-45.4Ph 1Terminated1Nov 20231results
NCT05158244Study of Multiple Oral Doses of PF-07081532 in Adult Participants With Type 2 Diabetes Mellitus

Lotiglipron

Obesity / overweight, Type 2 diabetes

BMI 24.5-45.5Ph 1Completed1Jun 20221results
NCT05788328A Drug-Drug Interaction Study to Estimate the Effect of PF-07081532 on the Pharmacokinetics of Dabigatran and Rosuvastatin in Overweight or Obese Adult Participants

Lotiglipron

Healthy volunteers, Obesity / overweight

BMI ≥25Ph 1Terminated1Sep 20231results
NCT05745701A Drug-Drug Interaction Study to Examine the Impact of Itraconazole and Cyclosporine on PF-07081532 Pharmacokinetics in Overweight or Obese Adults

Lotiglipron

Obesity / overweight

BMI ≥25Ph 1Completed1May 2023results
NCT05677867A Study to Compare Two Different Forms of PF-07081532 in Adults Who Are Overweight or Obese

Lotiglipron

Obesity / overweight

BMI 25-34.9Ph 1Completed1Mar 2023results
NCT05652647A Study to Understand How the Study Medicine (PF-07081532) is Processed and Eliminated in Healthy Men

Lotiglipron

Healthy volunteers

BMI 17.5-30.5Ph 1Completed1Mar 2023results
NCT04148209Study of Single Ascending Doses of PF-07081532 in Healthy Adult Participants

Lotiglipron

Healthy volunteers

BMI 17.5-30.5Ph 1Completed1Mar 2020